Search Result "imidazoacridinones"


Mechanisms of Action of Imidazoacridinone and Triazoloacridinone Derivatives in View of their Biological Activity

Journal: Current Pharmaceutical Analysis
Volume: 7 Issue: 4 Year: 2011 Page: 286-295
Author(s): Marcin Koba, Tomasz Baczek

Influence of LC Retention Data on Antitumor Acridinones’ Classification Evaluated by Factor Analysis Method

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 15 Issue: 8 Year: 2012 Page: 674-683
Author(s): Marcin Koba,Tomasz Baczek,Tomasz Ciesielski

The Application of Connected QSRR and QSAR Strategies to Predict the Physicochemical Interaction of Acridinone Derivatives with DNA

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 17 Issue: 10 Year: 2014 Page: 820-826
Author(s): Paulina Szatkowska-Wandas,Marcin Koba,Agata Kuchcicka,Sylwia Kurek,Emilia Daghir-Wojtkowiak,Tomasz Baczek

Application of Artificial Neural Networks for the Prediction of Antitumor Activity of a Series of Acridinone Derivatives

Journal: Medicinal Chemistry
Volume: 8 Issue: 3 Year: 2012 Page: 309-319
Author(s): Marcin Koba

The Influence of Lipophilicity on the Classification of Antitumor Acridinones Evaluated by Principal Component Analysis

Journal: Current Pharmaceutical Analysis
Volume: 8 Issue: 2 Year: 2012 Page: 157-174
Author(s): Marcin Koba,Tomasz Baczek

Chemometric Evaluation of the Significance of Molecular Structural Descriptors on Binding of Acridinone Derivatives to DNA

Journal: Letters in Drug Design & Discovery
Volume: 7 Issue: 7 Year: 2010 Page: 494-499
Author(s): Marcin Koba, Tomasz Baczek

Prediction of Acridinones’ Ability to Interstrand DNA Crosslinks Formation Using Connected QSRR and QSAR Analysis

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 5 Year: 2016 Page: 387-394
Author(s): Paulina Szatkowska-Wandas,Marcin Koba

The Evaluation of Multivariate Adaptive Regression Splines for the Prediction of Antitumor Activity of Acridinone Derivatives

Journal: Medicinal Chemistry
Volume: 9 Issue: 8 Year: 2013 Page: 1041-1050
Author(s): Marcin Koba,Tomasz Bączek

Is DNA Minor Groove Binding Crucial for Biological Activity of Triazoloacridinones with Cytotoxic and Antitumour Properties?

Journal: Letters in Drug Design & Discovery
Volume: 6 Issue: 4 Year: 2009 Page: 242-245
Author(s): Marcin Koba, Katarzyna Koba, Tomasz Baczek

Review Article

Nanostructured Systems for the Organelle-specific Delivery of Anticancer Drugs

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 224-236
Author(s): Graziella Anselmo Joanitti,Rayane Ganassin,Mosar Correa Rodrigues,Joao Paulo Figueiro Longo,Cheng-Shi Jiang,Jinsong Gu,Sandra Milena Leal Pinto,Maria de Fatima Menezes Almeida dos Santos,Ricardo Bentes de Azevedo,Luis Alexandre Muehlmann

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